Biomolecules & Therapeutics : eISSN 2005-4483 / pISSN 1976-9148

Table. 1.

EC50 values of GPR43 agonists

EC50 (μM)
cAMP Ca2+ β-Arrestin 2 NF-κB
Acetate 300.7 57.72 1,438 77.38
PAAT 0.089 7.673 4.15 12.06
Compound 110 18.65 2.410 1.609 3.406
Compound 187 0.016 0.019 0.018 0.019
Biomolecules & Therapeutics 2022;30:48~54 https://doi.org/10.4062/biomolther.2021.078
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