Biomolecules & Therapeutics : eISSN 2005-4483 / pISSN 1976-9148

Cited by CrossRef (32)

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  12. Kyeong-Man Kim. Conceptual Progress for the Improvements in the Selectivity and Efficacy of G Protein-Coupled Receptor Therapeutics: An Overview. Biomolecules & Therapeutics 2017;25:1
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  13. Leif Hertz, Ye Chen. Glycogenolysis, an Astrocyte-Specific Reaction, is Essential for Both Astrocytic and Neuronal Activities Involved in Learning. Neuroscience 2018;370:27
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  15. Liang Tan, Wenzhong Yan, John D. McCorvy, Jianjun Cheng. Biased Ligands of G Protein-Coupled Receptors (GPCRs): Structure–Functional Selectivity Relationships (SFSRs) and Therapeutic Potential. J. Med. Chem. 2018;61:9841
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  16. Xiaofei E, Paul Meraner, Ping Lu, Jill M. Perreira, Aaron M. Aker, William M. McDougall, Ronghua Zhuge, Gary C. Chan, Rachel M. Gerstein, Patrizia Caposio, Andrew D. Yurochko, Abraham L. Brass, Timothy F. Kowalik. OR14I1 is a receptor for the human cytomegalovirus pentameric complex and defines viral epithelial cell tropism. Proc Natl Acad Sci USA 2019;116:7043
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  17. Jolien Storme, Dilip K. Tosh, Zhan-Guo Gao, Kenneth A. Jacobson, Christophe P. Stove. Probing structure-activity relationship in β-arrestin2 recruitment of diversely substituted adenosine derivatives. Biochemical Pharmacology 2018;158:103
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  18. Supachoke Mangmool, Warisara Parichatikanond, Hitoshi Kurose. Therapeutic Targets for Treatment of Heart Failure: Focus on GRKs and β-Arrestins Affecting βAR Signaling. Front. Pharmacol. 2018;9
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  20. Yusuke Shintani, Atsuko Hayata-Takano, Keita Moriguchi, Takanobu Nakazawa, Yukio Ago, Atsushi Kasai, Kaoru Seiriki, Norihito Shintani, Hitoshi Hashimoto, Arun Shukla. β-Arrestin1 and 2 differentially regulate PACAP-induced PAC1 receptor signaling and trafficking. PLoS ONE 2018;13:e0196946
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  21. Teja Devarakonda, Fadi N. Salloum. Heart Disease and Relaxin: New Actions for an Old Hormone. Trends in Endocrinology & Metabolism 2018;29:338
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  23. Jingwei Bian, Suli Zhang, Ming Yi, Mingming Yue, Huirong Liu. The mechanisms behind decreased internalization of angiotensin II type 1 receptor. Vascular Pharmacology 2018;103-105:1
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  26. Mohammad Golam Sabbir, Paul Fernyhough. Muscarinic receptor antagonists activate ERK-CREB signaling to augment neurite outgrowth of adult sensory neurons. Neuropharmacology 2018;143:268
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  27. Valerie T. Ramirez, Wesley E. P. A. van Oeffelen, Cristina Torres-Fuentes, Barbara Chruścicka, Clementine Druelle, Anna V. Golubeva, Marcel van de Wouw, Timothy G. Dinan, John F. Cryan, Harriët Schellekens. Differential functional selectivity and downstream signaling bias of ghrelin receptor antagonists and inverse agonists. The FASEB Journal 2019;33:518
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  28. Cristina Torres-Fuentes, Elena Pastor-Cavada, Rafael Cano, Dalia Kandil, Rachel Shanahan, Rocio Juan, Hamdy Shaban, Gerard McGlacken, Harriët Schellekens. Quinolones Modulate Ghrelin Receptor Signaling: Potential for a Novel Small Molecule Scaffold in the Treatment of Cachexia. IJMS 2018;19:1605
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  29. Shaherin Basith, Minghua Cui, Stephani J. Y. Macalino, Jongmi Park, Nina A. B. Clavio, Soosung Kang, Sun Choi. Exploring G Protein-Coupled Receptors (GPCRs) Ligand Space via Cheminformatics Approaches: Impact on Rational Drug Design. Front. Pharmacol. 2018;9
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  30. Hideaki Kanki, Tsutomu Sasaki, Shigenobu Matsumura, Satoru Yokawa, Toshiro Yukami, Munehisa Shimamura, Manabu Sakaguchi, Tadahide Furuno, Takahiro Suzuki, Hideki Mochizuki. β-arrestin-2 in PAR-1-biased signaling has a crucial role in endothelial function via PDGF-β in stroke. Cell Death Dis 2019;10
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  31. Ichio Shimada, Takumi Ueda, Yutaka Kofuku, Matthew T. Eddy, Kurt Wüthrich. GPCR drug discovery: integrating solution NMR data with crystal and cryo-EM structures. Nat Rev Drug Discov 2019;18:59
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  32. Chayma El Khamlichi, Flora Reverchon-Assadi, Nadège Hervouet-Coste, Lauren Blot, Eric Reiter, Séverine Morisset-Lopez. Bioluminescence Resonance Energy Transfer as a Method to Study Protein-Protein Interactions: Application to G Protein Coupled Receptor Biology. Molecules 2019;24:537
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